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OPTALIDON 500 mg/75 mg SUPPOSITORIES

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Prescription review online

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This page is for general information. Consult a doctor for personal advice. Call emergency services if symptoms are severe.
About the medicine

How to use OPTALIDON 500 mg/75 mg SUPPOSITORIES

Translated with AI

This page provides general information and does not replace a doctor’s consultation. Always consult a doctor before taking any medication. Seek urgent medical care if symptoms are severe.

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Introducción

Prospecto: información para el paciente

Optalidon 500 mg/75mg supositorios Propifenazona, cafeína anhidra

Lea todo el prospecto detenidamente antes de empezar a usar este medicamento, porque contiene información importante para usted.

Siga exactamente las instrucciones de administración del medicamento contenidas en este prospecto o las indicadas por su médico o farmacéutico

  • Conserve este prospecto, ya que puede tener que volver a leerlo.
  • Si necesita consejo o más información, consulte a su farmacéutico.
  • Si experimenta efectos adversos, consulte a su médico o farmacéutico, incluso si se trata de efectos adversos que no aparecen en este prospecto. Ver sección 4.
  • Debe consultar a un médico si empeora o si no mejora después de 10 días

Contenido del prospecto

  1. Qué es Optalidon y para qué se utiliza
  2. Qué necesita saber antes de empezar a usar Optalidon
  3. Cómo usar Optalidon
  4. Posibles efectos adversos
  5. Conservación de Optalidon
  6. Contenido del envase e información adicional

1. Qué es Optalidon y para qué se utiliza

Optalidon? es un medicamento que contiene dos activos en asociación: propifenazona para el dolor, y cafeína que tiene tiene una acción estimulante del sistema nervioso, para la somnolencia.

Está indicado para adultos y niños mayores de 12 años, para el alivio del dolor leve o moderado, como dolor de cabeza, dolor dental y dolor menstrual.

Debe consultar a un médico si empeora o si no mejora después de 10 días.

Doctor consultation

Not sure if this medicine is right for you?

Discuss your symptoms and treatment with a doctor online.

2. Qué necesita saber antes de empezar a usar Optalidon

No useOptalidon

  • Si es alérgico a propifenazona o a la cafeína, o a alguno de los demás componentes de este medicamento (incluidos en la sección 6).
  • Si es alérgico a medicamentos que contienen metamizol, fenilbutazona u otros componentes del grupo de las pirazolonas.
  • Si alérgico a medicamentos que contienen aminofilina, diprofilina, oxtrifilina, teobromina, teofilina u otros componenets del grupo de las xantinas.
  • Si ha presentado reacciones alérgicas de tipo asmático (dificultad para respirar, ahogo, broncoespasmos y en algunos casos tos o pitidos al respirar) al tomar ácido acetilsalicílico o a otros antiinflamatorios no esteroideos.
  • Si sufre alteraciones sanguíneas (granulocitopenia, agranulocitosis).
  • Si padece alguna enfermedad metabólica como porfiria (trastorno raro, normalmente hereditario, en el que se elimina gran cantidad de porfirina en heces y orina) o déficit congénito de glucosa-6- fosfato-deshidrogenasa.
  • Si padece de enfermedad grave del hígado, riñón o corazón (insuficiencia renal, hepática o cardíaca).
  • Si tiene trastorno de ansiedad
  • Si padece úlcera gastroduodenal activa.

Advertencias y precauciones

Consulte a su médico o farmacéutico antes de empezar a usar Optalidon.

No exceder la dosis recomendada en el apartado de Posología, ni utilizarlo más de 10 días. Consulte a su médico farmacéutico antes de empezar a usar Optalidon si:

  • tiene hipertensión,
  • tiene úlcera gastroduodenal,
  • si padece asma o enfermedades respiratorias graves (enfermedad pulmonar obstructiva crónica, enfisema, bronquitis crónica

Si el dolor persiste, empeora o aparecen otros síntomas, especialmente fiebre o úlceras en la boca, se debe interrumpir inmediatamente el tratamiento y consultar con su médico.

La cafeína puede elevar los niveles de glucosa en sangre.

En personas con dificultades para dormir, se recomienda no tomar este medicamento en las horas previas a acostarse, para evitar el posible insomnio.

Se debe informar a los deportistas que este medicamento contiene un componente que puede establecer un resultado analítico de control del dopaje como positivo.

Niños y adolescentes

No debe administrarse a niños menores de 12 años.

Otros medicamentos y Optalidon

Toma de Optalidon con otros medicamentos.

Informe a su médico o farmacéutico si está tomando o utilizando, ha tomado o utilizado recientemente o pudiera tener que tomar o utilizar cualquier otro medicamento. En particular, si está tomando alguno de los siguientes medicamentos, puede ser necesario modificar la dosis de alguno de ellos o la interrupción del tratamiento:

  • anticoagulantes orales (medicamentos que se utilizan para “fluidificar” la sangre y evitar la aparición de coágulos) como warfarina,
  • barbitúricos (medicamentos utilizados para el tratamiento de las convulsiones),
  • antihistamínicos (utilizados para reducir los síntomas de las reacciones alérgicas),
  • litio (disminuyendo su efecto terapéutico)

Uso de Optalidon con alimentos y bebidas y alcohol

Se recomienda limitar el uso de productos que contengan cafeína cuando se esté en tratamiento con este medicamento.

Embarazo y lactancia y fertilidad

Si está embarazada o en periodo de lactancia, cree que podría estar embarazada o tiene intención de quedarse embarazada, consulte a su médico o farmacéutico antes de utilizar este medicamento. No debe tomarse este medicamento durante el embarazo ni la lactancia sin consultar al médico.

No tome Optalidon si está en los últimos 3 meses de embarazo, ya que podría dañar al feto o causar problemas en el parto. Puede causar problemas renales y cardíacos en el feto. Puede afectar su tendencia y la del feto a sangrar y hacer que el trabajo de parto sea más tarde o más largo de lo esperado. No debe tomar Optalidon durante los primeros 6 meses de embarazo a menos que sea absolutamente necesario y lo indique su médico. Si necesita tratamiento durante este período o mientras está tratando de quedarse embarazada, se debe usar la dosis más baja durante el menor tiempo posible. Si se toma durante más de unos pocos días a partir de las 20 semanas de embarazo, Optalidon puede causar problemas renales en el feto que pueden provocar niveles bajos de líquido amniótico que rodea al feto (oligohidramnios) o estrechamiento de un vaso sanguíneo (ductus arteriosus) en el corazón del bebé. Si necesita tratamiento durante más días, su médico puede recomendar un control adicional.

Conducción y uso de máquinas

No conduzca ni maneje maquinaria peligrosa ya que este medicamento produce somnolencia o disminución de la capacidad de reacción a las dosis recomendadas.

3. Cómo usar Optalidon

Siga exactamente las instrucciones de administración de este medicamento indicadas por su médico o farmacéutico. En caso de duda, consulte de nuevo a su médico o farmacéutico.

Vía rectal.

La dosis recomendada es de 1 supositorio al día. La dosis máxima será de 2 supositorios día.

Debe utilizar siempre la dosis menor que sea efectiva. La administración del preparado está supeditada a la aparición del dolor. A medida que éste desaparezca debe suspenderse esta medicación.

Instrucciones para la correcta administración del preparado

Si el supositorio está demasiado blando para insertarlo, enfríelo en la nevera durante 30 minutos o póngalo bajo el chorro de agua fría antes de quitar la envoltura plástica o después si fuera necesario para evitar su reblandecimiento.

Uso en niños y adolescentes

No se debe utilizar en niños menores de 12 años.

Si usa más Optalidon del que debe

Los síntomas por sobredosis son: dolor abdominal, náuseas, vómitos, somnolencia, excitación, convulsiones y coma.

En caso de sobredosis o ingestión accidental, acudir inmediatamente a un centro médico o llamar al Servicio de Información Toxicológica (Teléfono: (91)-562.04.20), indicando el medicamento y la cantidad ingerida.

Si olvidó usar Optalidon

No use una dosis doble para compensar las dosis olvidadas.

Si interrumpe el tratamiento con Optalidon

Si tiene cualquier otra duda sobre el uso de este medicamento, pregunte a su médico o farmacéutico.

Medicine questions

Started taking the medicine and have questions?

Discuss your symptoms and treatment with a doctor online.

4. Posibles efectos adversos

Al igual que todos los medicamentos, este medicamento puede producir efectos adversos, aunque no todas las personas los sufran.

No suelen observarse a las dosis recomendadas. En sujetos hipersensibles se han observado muy raramente reacciones alérgicas de tipo cutáneo: enrojecimiento o picor, alteraciones en la piel con formación de ampollas, urticaria o shock. En este caso, interrumpir el tratamiento y acudir al médico. Ocasionalmente pueden aparecer mareos, náuseas, nerviosismo, dificultad para dormir, latidos cardíacos rápidos o irritación gastrointestinal.

Comunicación de efectos adversos

Si experimenta cualquier tipo de efecto adverso, consulte a su médico o farmacéutico, incluso si se trata de posibles efectos adversos que no aparecen en este prospecto. También puede comunicarlos directamente a través del Sistema Español de Farmacovigilancia de Medicamentos de Uso Humano: www.notificaram.es.

Mediante la comunicación de efectos adversos usted puede contribuir a proporcionar más información sobre la seguridad de este medicamento.

5. Conservación de Optalidon

Mantener este medicamento fuera de la vista y del alcance de los niños. No se requieren condiciones especiales de conservación.

No utilice este medicamento después de la fecha de caducidad que aparece en la etiqueta y en la caja después de CAD. La fecha de caducidad es el último día del mes que se indica.

Los medicamentos no se deben tirar por los desagües ni a la basura. Deposite los envases y los medicamentos que no necesita en el Punto SIGRE de la farmacia. Pregunte a su farmacéutico cómo deshacerse de los envases y de los medicamentos que ya no necesita. De esta forma, ayudará a proteger el medio ambiente.

6. Contenido del envase e información adicional

Composición de Optalidon

Por supositorio:

Los principios activos son propifenazona (DCI) 500 mg, cafeína anhidra 75 mg.

Los demás componentes (excipientes) son óxido de hierro amarillo, óxido de hierro rojo, Sorbitan laurato (Span 20) y masa para supositorios.

Aspecto del producto y contenido del envase

Envase con 6 supositorios.

Titular de la autorización de comercialización

Perrigo España S.A

Pza de Xavier Cugat 2 Edificio D planta 1 08174 Sant Cugat del Valles

Barcelona España

Responsable de la fabricación

MIPHARM. S.PA,

Via B. Ouaranta, 12, 1-201 40, Italia

Fecha de la última revisión de este prospecto: 12/2022

Otras fuentes de información

La información detallada de este medicamento está disponible en la página web de la Agencia Española de Medicamentos y Productos Sanitarios (AEMPS) http://www.aemps.gob.es

Online doctors for OPTALIDON 500 mg/75 mg SUPPOSITORIES

Discuss questions about OPTALIDON 500 mg/75 mg SUPPOSITORIES, including use, safety considerations and prescription review, subject to medical assessment and local regulations.

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Hocine Lokchiri

General medicine 21 years exp.

Dr. Hocine Lokchiri is a French consultant with over 20 years of experience in General and Emergency Medicine. He works with adults and children, helping patients with urgent symptoms, infections, sudden health changes and everyday medical concerns that require timely evaluation. His background includes clinical practice in France, Switzerland and the United Arab Emirates, which allows him to navigate different healthcare systems and manage a wide range of conditions with confidence. Patients value his calm, structured approach, clear explanations and evidence-based decision-making.

Online consultations with Dr. Lokchiri are suitable for many situations when someone needs quick medical guidance, reassurance or a clear next step. Common reasons for booking include:

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Many patients reach out when symptoms appear suddenly and cause concern, when a child becomes unwell unexpectedly, when a rash changes or spreads, or when it’s unclear whether an in-person examination is necessary. His emergency medicine background is particularly valuable online, helping patients understand risk levels, identify warning signs and choose safe next steps.

Some situations are not suitable for online care. If a patient has loss of consciousness, severe chest pain, uncontrolled bleeding, seizures, major trauma or symptoms suggesting a stroke or heart attack, he will advise seeking immediate local emergency services. This improves safety and ensures patients receive the right level of care.

Dr. Lokchiri’s professional training includes:

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He is an active member of several professional organisations, including the French Society of Emergency Medicine (SFMU), the French Association for Emergency Physicians (AMUF) and the Swiss Society of Emergency and Rescue Medicine (SGNOR). In consultations, he works with clarity and precision, helping patients understand their symptoms, possible risks and the safest treatment options.
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Chikeluo Okeke

General medicine 4 years exp.

Dr Chikeluo Okeke is an internal medicine doctor with extensive international clinical experience. Originally from Nigeria, he has worked across multiple European healthcare systems and currently practises in Sweden. This professional path has given him a strong understanding of different medical approaches and the ability to work effectively with patients from diverse cultural and linguistic backgrounds.

Dr Okeke focuses on general internal medicine and adult primary care, combining clinical accuracy with careful attention to lifestyle, personal context, and everyday health concerns. His consultations are particularly well suited for people who seek medical advice online, live abroad, or need clear guidance without unnecessary complexity.

He provides online consultations covering symptom assessment, prevention, and long-term management of chronic conditions, helping patients understand what is happening and decide on appropriate next steps.

Common reasons for consultation:

  • General internal medicine concerns and initial health assessment.
  • Acute symptoms such as fever, cough, infections, pain, or weakness.
  • Chronic conditions and treatment adjustment.
  • Blood pressure issues, fatigue, metabolic concerns.
  • Preventive consultations and routine check-ups.
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Dr Okeke is known for his clear communication, calm approach, and cultural awareness. He listens carefully, explains medical decisions in a structured way, and supports patients in making informed choices about their health.

Online consultations with Dr Chikeluo Okeke offer reliable internal medicine care without geographic limitations, focused on medical relevance, clarity, and patient comfort.

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Andrei Popov

General medicine 7 years exp.

Dr. Andrei Popov is a family physician with specialized training in the management of chronic pain. He provides video consultations for adults in Spain and across Europe: whether you have been living with pain for months that no one has been able to properly explain, or you need to resolve a health issue without waiting weeks for an appointment.

His approach is clear: to listen, organize your case, and provide you with a practical roadmap based on evidence-based medicine and adapted to your medical history and personal needs.

Pain: how he can help

  • Chronic pain (more than 3 months
  • Migraine and recurrent or high-intensity headaches
  •  Neck, lower back, back and joint pain
  •  Post-traumatic pain after injuries or surgeries
  •  Pain of neurological origin: neuralgia, neuropathic pain, fibromyalgia

General medicine

  • Frequent respiratory infections (cold, flu, persistent cough)
  • Hypertension, diabetes and metabolic disorders
  • Review of laboratory tests and MRI/CT reports (explained in clear language)
  • Preventive medicine and health monitoring
  • Second opinions and treatment adjustments (when clinically appropriate)

What the consultation is like
 Each session lasts up to 30 minutes. We review symptoms, medical history, medications and any tests you provide, and you finish the consultation with a clear treatment plan, defined next steps, and criteria to understand when follow-up may be needed. If warning signs are detected, he will clearly advise whether you need in-person care or urgent medical attention.

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Doctor

Yevgen Yakovenko

General surgery 12 years exp.

Dr. Yevgen Yakovenko is a licensed surgeon and general practitioner in Spain and Germany. He specialises in general, paediatric, and oncological surgery, internal medicine, and pain management. He offers online consultations for adults and children, combining surgical precision with therapeutic support. Dr Yakovenko works with patients across different countries and provides care in Ukrainian, Russian, English, and Spanish.

Areas of medical expertise:

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Experience and qualifications:

  • 12+ years of clinical experience in university hospitals in Germany and Spain.
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Doctor

Joao Silva

General medicine 6 years exp.

Dr. João Silva is a physician with training and experience in the field of General and Family Medicine, dedicated to providing healthcare focused on the well-being and quality of life of his patients. Throughout his professional career, he has developed broad clinical competencies, striving to maintain a medical practice based on scientific evidence and continuous knowledge updates.

Between 2013 and 2019, he completed the Integrated Master's Degree in Medicine at the Abel Salazar Institute of Biomedical Sciences in Porto, where he acquired a solid academic and clinical education.

Subsequently, between January 2021 and December 2021, he completed the General Internship at the Entre Douro e Vouga Hospital Center in Santa Maria da Feira, where he had the opportunity to work in different hospital settings and deepen his competencies in several areas of medicine.

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Complementing his medical training, Dr. João Silva also completed a Postgraduate Degree in Continuing and Palliative Care at CESPU, strengthening his preparation in the comprehensive approach to patient care, especially in situations requiring prolonged care and multidisciplinary support.

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€55
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Bulat Garipov

General medicine 15 years exp.

Dr. Bulat Garipov is a radiologist with more than 15 years of experience, specializing in magnetic resonance imaging (MRI). Throughout his professional career, he has worked in leading diagnostic imaging centers, both in on-site practice and teleradiology, which has allowed him to develop a broad and versatile approach to radiology.

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Additionally, Dr. Garipov is open to new collaboration opportunities in radiology and teleradiology projects. He offers his expertise in MRI, providing both first and second readings of studies, as well as advanced image interpretation, ensuring accurate and high-quality diagnostics.

You could consult Dr. Bulat Garipov in cases where accurate interpretation of MRI studies or a second expert opinion is required. His expertise is especially valuable in cases of suspected neurological conditions, back and joint pain, vascular disorders, as well as in the diagnosis of abdominal and pelvic diseases. The doctor also provides support in complex or unclear clinical situations, including the review of previously performed studies, which helps improve diagnostic accuracy and determine the optimal treatment strategy. A teleradiology format is available, allowing you to receive a professional opinion remotely.

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Frequently Asked Questions

Is a prescription required for OPTALIDON 500 mg/75 mg SUPPOSITORIES?
OPTALIDON 500 mg/75 mg SUPPOSITORIES does not require a prescription in Spain. You can check with a doctor online whether this medicine may be appropriate for your situation.
What is the active substance in OPTALIDON 500 mg/75 mg SUPPOSITORIES?
The active ingredient in OPTALIDON 500 mg/75 mg SUPPOSITORIES is propyphenazone, combinations excl. psycholeptics. This information helps identify medicines with the same composition but different brand names.
Who manufactures OPTALIDON 500 mg/75 mg SUPPOSITORIES?
OPTALIDON 500 mg/75 mg SUPPOSITORIES is manufactured by Perrigo Espana S.A.. Pharmacy brands and packaging may differ depending on the distributor.
Which doctors can assess the use of OPTALIDON 500 mg/75 mg SUPPOSITORIES online?
Doctors such as Family doctors, Psychiatrists, Dermatologists, Cardiologists, Endocrinologists, Gastroenterologists, Pulmonologists, Nephrologists, Rheumatologists, Hematologists, Infectious disease physicians, Allergists, Geriatricians, Paediatricians, Oncologists may assess whether OPTALIDON 500 mg/75 mg SUPPOSITORIES is appropriate, depending on your situation and local regulations. You can book an online consultation to discuss your symptoms and possible next steps.
What are the alternatives to OPTALIDON 500 mg/75 mg SUPPOSITORIES?
Other medicines with the same active substance (propyphenazone, combinations excl. psycholeptics) include METALGIAL 500 MG/ML ORAL DROPS IN SOLUTION, METAMIZOLE ABABOR 575 mg HARD CAPSULES, METAMIZOL AIKO FARMACEUTICA 575 mg HARD CAPSULES. These may have different brand names or formulations but contain the same therapeutic ingredient. Always consult a doctor before switching or starting a new medicine.
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